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Degrader-Drug Conjugate (DDC) Mediated Immunochemotherapy for Tumor Treatment

J. Med. Chem. 2025, https://doi.org/10.1021/acs.jmedchem.5c02262

12. Chaoming Wang,Jing Zhang, Dongping Wang, Shengle Chen, Qi Yuan, Ruijuan Yin, Guiyang Yao, Xin Qi, Jing Li*, and Tao Jiang*

Conjugating 10,11-Dimethoxy-camptothecin with an Integrin αvβ3-Targeting Peptide through a Triazine Linker for Targeted Tumor

Treatment in Lung and Pancreatic Carcinoma

J. Med. Chem. 2025, 68, 23, 25091–25111 https://doi.org/10.1021/acs.jmedchem.5c02059

11. Yi Zhou , Jingyan Jin, Pingzheng Zhou*, Wu Su* , Guiyang Yao*

Adding A C-Terminal Amino Acid Prevents the Conformational Interconversion of Plecantide Analogs

ChemBioChem 2025, 26, e202500237. (Front cover, The 18th Chinese International Peptide Symposium)

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 Computationally Designed Epitope-Mediated Imprinted Polymers versus Conventional Epitope Imprints for the Detection of Human Adenovirus in Water and Human Serum Samples. 

ACS sensors, 2024, https://doi.org/10.1021/acssensors.3c02374

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The occurrence of ansamers in the synthesis of cyclic peptides.

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Iodine-Mediated Tryptathionine Formation Facilitates the Synthesis of Amanitins.

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Nitidumpeptins A and B, Cyclohexapeptides Isolated from Zanthoxylum nitidum var. tomentosum: Structural Elucidation, Total Synthesis, and Antiproliferative Activity in Cancer Cells.

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Novel N-Methylated Cyclodepsipeptide Prodrugs for Targeted Cancer Therapy.

J Med Chem 2021 64, 991-1000. 10.1021/acs.jmedchem.0c01387      

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Total Synthesis of the Death Cap Toxin Phalloidin: Atropoisomer Selectivity Explained by Molecular-Dynamics Simulations.

Chem.-Eur. J. 2019, 25, 8030– 8034.https://chemistry-europe.onlinelibrary.wiley.com/doi/abs/10.1002 /chem.201901888   

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Improved total synthesis and biological evaluation of coibamide A analogues. 

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N-terminal α-amino group modification of antibodies using a site-selective click chemistry method. 

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Efficient Synthesis and Stereochemical Revision of Coibamide A.

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Fully Automated Synthesis of DNA-Binding Py-Im Polyamides Using a Triphosgene Coupling Strategy. 

Org. Lett. 2014, 17, 158-161. https://pubs.acs.org/doi/abs /10.1021/ol503388a